Bayoumi, A. H. Antiproliferative Properties of Vinyl Dipeptides: Synthesis and MCF-7 Cell Line Testing. 2012.
Mousa, B. A.; Bayoumi, A. H.; Korraa, M. M.; Assy, M. G.; El-kalyoubi, S. A. Synthesis, DNA binding studies of new pyrimidothiazepine and pyrimidobenzothiazepine derivatives. Afinidad 2012, 69.
Synthesis and Anxiolytic Activity of Some Novel 5-oxo-1, 4-oxazepine Derivatives. Bothiana A. AbdelFattah, Maha M.A. Khalifa, Hend El-Sehrawi, Eman Fayed, Ashraf Bayoumi and Makarem Said. Letters in Drug Design & Discovery, 2011, 8, 330-338.
Synthesis and anticonvulsant evaluation of some new quinoxalinone derivatives. Ashraf Bayoumi, Adel Ghiaty, Ahmed El-Morsy, Hamada Abul-Khair and Salwa Elmeligie, Egypt. J. Biomed. Sci. Vol. 37, November 2011.
A Novel Method for Synthesis of Tertiary Benzamides Utilizing NBS. Ashraf Bayoumi. Egypt. J. Biomed. Sci. Vol. 37, November 2011.
Synthesis and evaluation of some new 1,2,4-triazolo(4,3-a)quinoxalin-4-5H-one derivatives as AMPA receptor antagonists. Ashraf Bayoumi, Adel Ghiaty, Ahmed El-Morsy, Hamada Abul-Khair, Memy H. Hassan, Salwa Elmeligie. Bulletin of Faculty of Pharmacy, Cairo University (2012) 50, 141–146.
Synthesis and preliminary antimicrobial evaluation of some new 6-methoxyquinoline-3- carbonitrile derivatives, Mohamed Hagrs a , Ashraf H. Bayoumi a , Kamal M. El-Gamal a,b , Abdelrahman S. Mayhoub a , Hamada S. Abulkhai, beni-suef university journal of basic and applied sciences 4 (2015) 338–345.
Synthesis of Pyrroles and Condensed Pyrroles as Anti-Inflammatory Agents with Multiple Activities and Their Molecular Docking Study, M. T. Sarg, M. M. Koraa, A. H. Bayoumi, S. M. Abd El Gilil, Open Journal of Medicinal Chemistry, 2015, 5, 49-96.
A Novel One-Pot and Efficient Procedure for Synthesis of New Fused Uracil Derivatives for DNA Binding, Bothaina A. Mousa1, Ashraf H. Bayoumi, Makarem M. Korraa1, Mohamed G. Assy, Samar A. El-Kalyoubi, International Journal of Organic Chemistry, 2015, 5, 37-47.
Design and Synthesis of Pyridine-amide Based Compounds Appended Naproxen Moiety as Anti-Microbial and Anti-inflammatory Agents, Yousry A. Ammar, Eman A. Fayed, Ashraf H. Bayoumi, Marwa A. Saleh, Moustafa E. El-Araby, Am. J. Pharm Tech Res. 2015; 5(6).
Synthesis and Biological Evaluation of New amides Pro-drugs Containing Naproxen Moiety as Anti-inflammatory and Antimicrobial Agents, Eman A. Fayed, Ashraf H. Bayoumi, Marwa A. Saleh, and Yousry A. Ammar, Der Pharma Chemica, 2016, 8(1):495-508.
Synthesis, reaction and antitumor screening of some new quinoline derivatives. Mohamed M. Ismail, Saber E.S. Barakat, Ashraf H. Bayomi, Helmy M. Sakr and Kamal M. A. El-Gamal. Department of Organic Chemistry, Faculty of Pharmacy, Cairo University, Cairo, Egypt, Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Al-Azhar University, Cairo, Egypt, Department of Organic Chemistry, Faculty of Pharmacy, AlAzhar University, Cairo, Egypt. Az. J. Pharm. Sci. Vol. 35 March, 104-111, 2007.
Synthesis, reaction and antitumor screening of some new quinoline and substituted 2-amino quinoline derivatives. Mohamed M. Ismail, Saber E.S. Barakat, Ashraf H. Bayomi, Helmy M. Sakr and Kamal M. A. ElGamal. Department of Organic Chemistry, Faculty of Pharmacy, Cairo University, Cairo, Egypt. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Al-Azhar University, Cairo, Egypt. Department of Organic Chemistry, Faculty of Pharmacy, Al-Azhar University, Cairo, Egypt. Az. J. Pharm. Sci. Vol. 36 September, 205-213, 2007.
Regioselective synthesis and antitumor screening of some novel N-phenylpyrazole derivatives. Ahmad M. Farag, Abdelrahman S. Mayhoub, Saber. Barakat and Ashraf H. Bayomi. Bioorg. Med. Chem. 16 (2008) 881-889
Synthesis of new N-phenylpyrazole derivatives with potent antimicrobial activity. Ahmad M. Farag, Abdelrahman S. Mayhoub, Saber E. Barakat and Ashraf H. Bayomi. Bioorg. Med. Chem. 16 (2008) 4569-4578.
Modeling, synthesis and antihyperglycemic activity of novel quinazolinones containing sulfonylurea moiety. Mohammed K. Ibrahim, Abd-Elghany A. El-Helby, Adel H. Ghiaty, Ashraf H. Bayoumi, Ashraf A. Abd-El Rahman, Rizk R. Ayya, Menshawy A. Menshawy, and Ibrahim H. Eissa. J. Biol. Pham. Sci. Vol. 7, No. 1 July, 2009.
Synthesis, anxiolytic activity and antimicrobial screening of some novel 5-oxo-1,4-oxazepine derivatives. Bothiana A. Abdel Fattah, Hend El-Sehrawi, Maha M.A. Khalifa, Eman Fayed, Ashraf Bayoumi and Makarem Said. Egypt. J. Biomed. Sci. Vol. 33, July, 2010.
Synthesis of 3-phenyl-4-(3H)-quinazolinone derivative as privileged templates and for biological screening. Bayomi, Ashraf Hassan. Organic Chemistry Department, Faculty of Pharmacy, Al-Azhar University, Nasr City, Egypt. Afinidad (2005), 62(517), 249-254
Synthesis of some New Dibenz[c,e]azepine-5,7-diones of Expected Antihyperlipidemic Activity. Saber ES. Barakat, Mohamed A.A. El-Zahaby, Ashraf A. Abdel-Rahman, Ashraf H. Bayomi*, Hany E. Ali* and Monir A-S. Amin, Pharmaceutical Chemistry Department and Organic Chemistry Department* Faculty of Pharmacy (Boys), Al-Azhar University, Nasr City, Cairo, Egypt. Egypt. J. Biomed. Sci. Vol. 19, 69-82, 2005.
Synthesis of some New 4(3H)Quinazolinone Derivatives for Biological Screening. El-Helby, Abdel-Ghany A.; Abdel Rahman, Ashraf. A; Bayomi, Ashraf H.; Zayed, Mohamed F. Pharmaceutical Chemistry Department, Faculty of Pharmacy, Al-Azhar University, Nasr City, Cairo-Egypt. 8th ICCRD Mansoura & Sharm El-Sheikh, April 11-14, 2005. PC-32.
Synthesis and antimicrobial activity of some new quinoline and 1H-pyrazolo[3,4-b]quinoline derivatives. Amin, Monir A.-S.; Ismail, Mohammed M.; Barakat, Saber E.-S.; Abdul-Rahman, Ashraf A.-A.; Bayomi, Ashraf H.; El-Gamal, Kamal M. A. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Al-Azhar University, Cairo, Egypt. Bulletin of Pharmaceutical Sciences, Assiut University (2004), 27(2), 237-245.
Synthesis and Preliminary Pharmacological Study of some New Derivatives of 1-Pheny-4oxo(1H)pyrazolo[3,4-d]pyrimidine Derivatives. Amin, Monir A.; Ismail, Mohamed M.; El-Helby, Abdel-Ghani A.; Bauomy, Ashraf H.; El-Morsy, Ahmed M. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, AlAzhar University, Nasr City, Cairo, Egypt and Department of Organic Chemistry, Faculty of Pharmacy, Cairo University, Cairo, Egypt. Alex. J. Pharm. Sci., Vol. 17(1), March, 1-11, 2003.
Vitamin B12 as carrier for anticancer drugs. Bayomi, Ashraf H.; Mitchell, Alice M.; Natarajan, Ettaya N.; Grissom, Charles B.; West, F. G.; Aziza, Mohsen A.; El-Ahmady, Omar. Department Chemistry, University Utah, Salt Lake City, UT, USA. Book of Abstracts, 214th ACS National Meeting, Las Vegas, NV, September 7-11 (1997), MEDI-123. Publisher: American Chemical Society, Washington, D. C
Triggered release of chlorambucil from an inactive bioconjugate. Bayomi, Ashraf H.; Mitchell, Alice M.; Natarajan, Ettaya N.; Grissom, Charles B.; West, F. G.; Aziza, Mohsen A.; El-Ahmady, Omar. Department of Chemistry, University of Utah, Salt Lake City, UT, USA. Book of Abstracts, 213th ACS National Meeting, San Francisco, April 13-17 (1997), MEDI-123. Publisher: American Chemical Society, Washington, D. C.
Sonolysis Promotes Indirect Co-C Bond Cleavage of Alkylcob(III)alamin Bioconjugates. Howard, W. Allen ,Jr.; Bayomi, Ashraf; Natarajan, Ettaya; Aziza, Mohsen A.; El-Ahmady, Omar; Grissom, Charles B.; West, Frederick G. Department of Chemistry, University of Utah, Salt Lake City, UT, USA. Bioconjugate Chemistry (1997), 8(4), 498-502.
Yehia, E.; Mohammad, H.; Abdelghany, M. T.; Fayed, I.; Seleem, M.; Mayhoub, A. S.* Phenylthiazole Antibiotics: A Metabolism Guided Approach to Overcome Short Duration of Action (2016). E. J. Med. Chem.
Eissa, I. H.; Mohammad, H.; Qassem, O. A.; Younis, W.; Abdelghany, T. M.; Elshafeey, A.; Moustafa, M. M. A. R.; Seleem, M. N.; Mayhoub, A. S. Diphenylurea derivatives for combating methicillin-and vancomycin-resistant Staphylococcus aureus. European Journal of Medicinal Chemistry 2017, 130, 73-85.
Mohammad, H.; Younis, W.; Chen, L.; Peters, C. E.; Pogliano, J.; Pogliano, K.; Cooper, B. R.; Zhang, J.; Mayhoub, A. S.; Oldfield, E. Phenylthiazole Antibacterial Agents Targeting Cell Wall Synthesis Exhibit Potent Activity In Vitro and In Vivo against Vancomycin-resistant Enterococci. J. Med. Chem. 2017.
Younis, W.; AbdelKhalek, A.; Mayhoub, A.; Seleem, M. In vitro screening of an FDA-Approved Library against ESKAPE pathogens. Curr. Pharm. Des. 2017.
Mohamed Hagras, Haroon Mohammad, Mohamed S. Mandour, Youssef A. Hegazy, Adel Ghiaty, Mohamed N. Seleem, and Abdelrahman S Mayhoub.* Investigating the Antibacterial Activity of Biphenylthiazoles against Methicillin- and Vancomycin-Resistant Staphylococcus aureus (MRSA and VRSA). J. Med. Chem. April 2017 (just accepted)
Farag, A. M.; Mayhoub, A. S.; Barakat, S. E.; and Bayomi, A. H. Regioselective Synthesis and Antitumor Screening of Some Novel N-Phenylpyrazole Derivatives. Bioorg. Med. Chem. 2008, 16, 881–889.
Farag, A. M.; Mayhoub, A. S.; Barakat, S. E.; and Bayomi, A. H. Synthesis of new N-Phenylpyrazole Derivatives with Potent Antimicrobial Activity. Bioorg. Med. Chem. 2008, 16, 4569–4578.
Shaaban, M. R.; Saleh, T. S.; Mayhoub, A. S.; Mansour, A.; and Farag, A. M. Synthesis and Analgesic/Anti-inflammatory Evaluation of Fused Heterocyclic Ring Systems Incorporating Phenylsulfonyl Moiety. Bioorg. Med. Chem. 2008, 16, 6344–6352.
Farag, A. M; Mayhoub, A. S.; El-Debss, T. M. A.; Amr, A. E.; Abdel-Hafez, N. A.; Ali, K. A. K.; and Abdulla, M. M. Synthesis and Structure-Activity Relationship Studies of Pyrazole-Based Heterocycles as Antitumor Agents. Arch. Pharm. Chem. Life Sci. 2010, 343, 384–396.
Mayhoub, A. S.; Talukdar, A.; Cushman, M. Oxidation of Benzyl Methyl Ethers with NBS Selectively Affords Either Aromatic Aldehydes or Aromatic Methyl Esters. J. Org. Chem. 2010, 75, 3507–3510.
Farag, A. M; Ali, K. A. K.; El-Debss, T. M. A.; Mayhoub, A. S.; Amr, A. E.; Abdel-Hafez, N. A.; and Abdulla, M. M. Design, Synthesis and Structure–Activity Relationship Study of Novel Pyrazole-Based Heterocycles as Potential Antitumor Agents. E. J. Med. Chem. 2010, 45, 5887–5898.
Mayhoub, A. S.; Kiselev, E.; Cushman, M. An Unexpected Synthesis of 3,5-Diaryl-1,2,4-Thiadiazoles from Thiobenzamides and Methyl Bromocyanoacetate. Tetrahedron Lett. 2011, 52, 4941–4943.
Mayhoub, A. S.; Khaliq, M.; Kuhn, R. J.; Cushman, M. Design, Synthesis, and Biological Evaluation of Thiazoles Targeting Flavivirus Envelope Proteins. J. Med. Chem. 2011, 54, 1704–1714.
Mayhoub, A. S.; Khaliq, M.; Z, Li; Kuhn, R. J.; Cushman, M. An Investigation of Phenylthiazle Antiflaviviral Agents. Bioorg. Med. Chem. 2011, 16, 3845–3854.
Shaaban, M. R..; Saleh, S. T.; Mayhoub, A. S.; and Farag, A. M. Single Step Synthesis of New Fused Pyrimidine Derivatives and Their Evaluation as Potent Aurora-A Kinase Inhibitors. E. J. Med. Chem. 2011, 46, 3690–3695.
Mayhoub, A. S.; Marler, L.; Kondratyuk, T.; Pezzuto, J. M.; Cushman, M. Optimization of Thiazole Analogues of Resveratrol for Induction of NAD(P)H:quinone Reductase 1 (QR1). Bioorg. Med. Chem. 2012, 20, 7030–7039.
Mayhoub, A. S.; Hepatitis C RNA-Dependent RNA Polymerase Inhibitors, A Review of Structure-Activity and Resistance Relationships Bioorg. Med. Chem. 2012, 20, 3150–3161.
Shaaban, M. R.; Mayhoub, A. S.; and Farag, A. M. Recent Advances in the Therapeutic Applications of Pyrazolines. Expert Opin. Ther. Pat. 2012, 22, 253–291.
Mayhoub, A. S.; Marler, L.; Kondratyuk, T.; Pezzuto, J. M.; Cushman, M. Optimization of the Aromatase Inhibitory Activities of Pyridylthiazole Analogues of Resveratrol. Bioorg. Med. Chem. 2012, 20, 2427–2434.
Marler, L.; Mayhoub, A. S.; Cushman, M.; Pezzuto, J. M. Thiazole and Thiadiazole Derivatives of Resveratrol as Inducers of Quinone Reductase 1. Pharm. Biol. 2012, 50, 541–541.
Mayhoub, A. S.; Marler, L.; Kondratyuk, T.; Pezzuto, J. M.; Cushman, M. 3,5-Optimization of Thiadiazole Analogues of Resveratrol vs. Three Chemopreventive Targets. Bioorg. Med. Chem. 2012, 20, 510–520.
Lu, J. W.; Xu, C.; Pei, Z.; Mayhoub, A. S.; Cushman, M.; Flockhart, D. A. The Tamoxifen metabolite Norendoxifen is a Potent and Selective Inhibitor of Aromatase (CYP19) and a Potential Lead Compound for Novel Therapeutic Agents. Breast Cancer Res. Treat. 2012,133, 99–109.
Pricer, R. E.; Houghton, J. L.; Green, K. D.; Mayhoub, A. S.; and Garneau-Tsodikova, S. Biochemical and Structural Analysis of Aminoglycoside Acetyltransferase Eis from Anabaena variabilis. Mol. BioSyst. 2012, 8, 3305–3313.
Eckroat, T. J.; Kochi, A.; Green, K. D.; Mayhoub, A. S.; Lim, M. H.; Garneau-Tsodikova, S. A Novel 6-Chlorotacrine-Metal Chelator Hybrid for Inhibition of Acetylcholinesterase and Prevention of Metal-Induced Amyloid-b Aggregation. Chem. Sci. 2013, 4, 4137–4145.
Eckroat, T.; Mayhoub, A. S.; Garneau-Tsodikova, S. Amyloid-β Probes: Review of Structure-Activity and Brain Kinetics Relationships Beilstein J. Org. Chem. 2013, 9, 1012–1044.
Houghton, J. L.; Green, K. D.; Pricer, R. E.; Mayhoub, A. S.; Garneau-Tsodikova, S. Unexpected N-Acetylation of Capreomycin by Mycobacterial Eis Enzymes. J. Antimicrob. Chemother. 2013, 68, 800–805.
Gomhaa, S. M.; Eldebss, T. A.; Abdullab, M. M.; Mayhoub, A. S. Diphenylpyrroles: Novel p53 Activators. E. J. Med. Chem. 2014, 82, 472–479.
Mohammad, H.; Mayhoub, A. S.; Ajlouni, R.; Cushman, M.; Seleem, M. Discovery and Characterization of Potent Thiazoles versus Methicillin- and Vancomycin-Resistant Staphylococcus aureus. J. Med. Chem. 2014, 57, 1609–1615.
Mohammad, H.; Reddy, P.V.; Mayhoub, A. S.; Cushman, M.; Hammac, G. K.; Seleem, M. Antibacterial characterization of Novel Synthetic Thiazole Compounds Against Methicillin-Resistant Staphylococcus pseudintermedius. PloS ONE, 2015, 10, e0130385.
Gomhaa, S. M.; Eldebss, T. A.; Badry, M. G.; Abdullab, M. M.; Mayhoub, A. S. Novel 4-Heteroaryl-Antipyrines as DPP-IV Inhibitors. Chem. Biol. Drug Des. 2015, 86, 1292–1303.
Badrey, M. G.; Gomha, S. M.; Abdalla, M. M.; Mayhoub, A. S. Design and Synthesis of Imidazopyrazolopyridines as Novel Selective COX-2 Inhibitors. Molecules 2015, 20, 15287–15303.
Mohammad, H.; Reddy, P.V.; Mayhoub, A. S.; Cushman, M.; Seleem, M. Synthesis and Antibacterial Evaluation of a Novel Series of Synthetic Phenylthiazole Compounds Against Methicillin-Resistant Staphylococcus aureus (MRSA). E. J. Med. Chem. 2015, 94, 306–316.
Mohammad, H.; Mayhoub, A. S.; Cushman, M.; Seleem, M. Anti-biofilm Activity and Synergism of Novel Thiazole Compounds with Glycopeptide Antibiotics Against Multidrug-Resistant Staphylococci. J. Antibiotics. 2015, 68, 259–266.
Seleem, M. A.; Disouky, A.; Mohammad, H.; Abdelghany, M. T.; Mancy, A. S.; Bayoumi. S. A.; Elshafeey, A.; El-Morsy, A.; Seleem, M.; Mayhoub, A. S.* Second-Generation Phenylthiazole Antibiotics with Enhanced Pharmacokinetic Properties. J. Med. Chem. 2016, 59, 4900–4912.
Kamal M. A. El-Gamal, Farag F. Sherbiny, Ahmed M. El-Morsi, Hamada S. Abulkhair, Ibrahim H. Eissa and Mohamed M. El-Sebaei. Synthesis, molecular docking and antimicrobial evaluation of some novel quinoline-3-carbaldehyde derivatives. Chem. Sci. Rev. Lett. 2015, 4, 1170-1187
Benjamin F. Seibt, Anke C. Schiedel, Dominik Thimm, Sonja Hinz, Farag F. Sherbiny, Astrid Maas and Christa E. Müller The second extracellular loop of GPCRs determines subtype-selectivity and controls efficacy as evidenced by loop exchange studies at A2 adenosine receptors. Biochemical Pharmacology 2013, 85, 1317-1329
Dominik Thimm, Anke C. Schiedel, Farag F. Sherbiny, Sonja Hinz, Katharina Hochheiser, Daniela C. G. Bertarelli, Astrid Maas and Christa E. Müller. Ligand-specific binding and activation of the human adenosine A2B receptor. Biochemistry 2013, 52, 726-740
Sonja Hinz, Anke C. Schiedel, Dominik Thimm, Farag Sherbiny, Thomas Borrmann, Astrid Maaß and Christa E. Müller One is all it takes: disulfide bonds and cysteine residues in the extracellular loop 2 of the adenosine A2B receptor. Abstracts of the Fourth Joint German-Italian Purine Club Meeting 2011 Purinergic Signalling 2012, 8, 174
Anke C. Schiedel, Sonja Hinza, Dominik Thimm, Farag Sherbiny, Thomas Borrmann, Astrid Maaß and Christa E. Müller The four cysteine residues in the second extracellular loop of the human adenosine A2B receptor: role in ligand binding and receptor function Biochem. Pharmacol. 2011, 82,389-399
Mohamed-Kamal Ibrahim, Ashraf A. Abd-Elrahman, Rezk R. A. Ayyad, Khaled El-Adl, Farag F Sherbiny and Mahmoud Rashed Design and synthesis of some novel N-phthalimide derivatives with potential anticonvulsant activity Az. J. Pharm. Sci. 2010, 42, 305-322
Anke Schiedel, Dominik T. Thimm, Sonja Hinz, Farag Sherbiny, Thomas Borrmann, Astrid Maaß and Christa E. Müller Importance of selected amino acid residues of the human adenosine A2B receptor for ligand binding and receptor activation. Purines 2010: Adenine Nucleosides and Nucleotides in Biomedicine. Purinergic Signal. 2010, 6, S36-S37
Anke C. Schiedel, Dominik Thimm, Sonja Hinz, Farag F. Sherbiny, Thomas Borrmann, Astrid Maaß and Christa E Müller Adenosine A(2B) receptors: Mutagenesis, modeling and new ligands to study drug-receptor interaction and activation. Third joint Italian-German Purine Club meeting: “Purinergic receptors: new frontiers for novel therapies” Purinergic signaling 2010, 6, 69
Farag F. Sherbiny, Anke C. Schiedel, Astrid Maaß, and Christa E. Müller Homology modelling of the human adenosine A2B receptor based on X ray structures of bovine rhodopsin, the β2-adrenergic receptor and the human adenosine A2A receptor J. Comput. Aided Mol. Des. 2009, 23, 807-828
A. A. El-Helby, M. A. Amin, M. M. El-Sawah, A. A. Bayomi, Adel S. El-Azab and Farag F. Sherbiny Synthesis and Microbiological Testing of Some new Derivatives of Compounds Containing Active Methylene Group J. Saudi Chem. Soc. 2006, 10, 77-94
Synthesis and Evaluation of Some New (1,2,4) Triazolo(4,3-a)Quinoxalin-4(5H)-one Derivatives as AMPA Receptor Antagonists, Hamada AbulKhair, Salwa Elmeligie, Ashraf Bayoumi, Adel Ghiaty, Ahmed El-Morsy, and Memy H. Hassan, Journal of Heterocyclic Chemistry, 50, 2013, 1202-1208.
Synthesis and anticonvulsant evaluation of some new quinoxalinone derivatives, Hamada Abulkhair, Salwa Elmeligie, Ashraf Bayoumi, Adel Ghiaty, Ahmed El-Morsy, and Memy H. Hassan, Egyptian Journal of Biomedical Sciences, 37, 2011, 46-58.
Synthesis and evaluation of some new 1,2,4-triazolo(4,3-a) quinoxalin-4-5H-one derivatives as AMPA receptor antagonists, Ashraf Bayoumi, Adel Ghiaty, Ahmed El-Morsy, Hamada Abulkhair, Memy H. Hassan, Salwa Elmeligie, Bulletin of Faculty of Pharmacy, Cairo University, 50, 2012, 141–146.
Synthesis, and antiviral evaluation of some new 2-(4-chlorophenyl)thiazole derivatives on yellow fever virus, Hamada Abulkhair, Al-Azhar Journal of Pharmaceutical Sciences Vol. 50, 2014, 255-266.
Synthesis and preliminary antimicrobial evaluation of some new 6-methoxyquinoline-3-carbonitrile derivatives, Mohamed Hagrs, Ashraf H. Bayoumi, Kamal M. El-Gamal, Abdelrahman S. Mayhoub, Hamada Abulkhair, Beni-suef University Journal of Basic and Applied Sciences, 4, 2015, 338–345.
Synthesis, molecular docking and antimicrobial evaluation of some novel quinoline-3-carbaldehyde derivatives, Kamal M. A. El-Gamal, Farag F. Sherbiny, Ahmad M. El-Morsi, Hamada Abulkhair, Ibrahim H. Eissa3 and Mohamed M. El-Sebaei, Chemical Science Review and Letters, 2015, 4(16), 1170-1187.
Synthesis, characterization and antimicrobial evaluation of some novel quinoline derivatives bearing different heterocyclic moieties, Kamal M. El-Gamal, Mohamed S. Hagrs, Hamada S. Abulkhair, Bulletin of Faculty of Pharmacy, Cairo University, 2016, 54(2), 263–273.
Molecular Docking, Synthesis and Biological Evaluation of Some Novel 2-Substituted-3-allyl-4(3H)-quinazolinone Derivatives as Anticonvulsant Agents, Hamada S. Abulkhair, Kamal M El-Gamal, Khaled El-Adl and Mohamed F Fadl, Medicinal Chemistry (Los Angeles), 2016, 6(9), 593-603
Ivanovich, R. A.; Vincent-Rocan, J.-F.; Elkaeed, E. B.; Andre M. Beauchemin, A. M. One-Pot Synthesis of Aza-Diketopiperazines Enabled by Controlled Reactivity of N‑Isocyanate Precursors. Org. Lett. 2015, 17, 4898-4901.
Elkaeed, E. B.; Ghiaty, A. H.; El-Morsy, A. M.; El-Gamal, K. A.; Sakr, H. Synthesis and Biological Evaluation of Some quinoxaline-2-one Derivatives as Novel Anticonvulsant Agents. Chem. Sci. Rev. Lett. 2014, 3(12), 1375-1387.
Younis, W.; AbdelKhalek, A.; Mayhoub, A. S. and Seleem, M. In vitro screening of an FDA-Approved Library against ESKAPE pathogens. Curr. Pharm. Des., 2017, 23, 1–11.
Yehia, E.; Mohammad, H.; Abdelghany, M. T.; Fayed, I.; Seleem, M.; Mayhoub, A. S.* Phenylthiazole Antibiotics: A Metabolism Guided Approach to Overcome Short Duration of Action Eur. J. Med. Chem. 2017, 126, 604–613.
Mohammad, H.; Younis, W.; Cooper, B.; Peters, C.E.; Pogliano, J. Pogliano, K.; Bruce, C.; Zhang, J.; A. S. Mayhoub, Oldfield, E.; Cushman, M.; Seleem. M. Phenylthiazole Antibacterial Agents Targeting Cell Wall Synthesis Exhibit Potent Activity in vitro and in vivo against Vancomycin-resistant Enterococci. J. Med. Chem. 2017, 60, 2425–2438.
Eissa, I., Mohammad, H.; Abdelghany, M. T.; Qassem, O. A., Younis, W.; Abdrabouh, M.; Seleem, M.; Mayhoub, A. S.* Diphenylurea Derivatives for Combating Methicillin- and Vancomycin-Resistant Staphylococcus aureus. Eur. J. Med. Chem. 2017, 130, 73–85.
Hagras, M.; Hegazy, Y.; Elkabbany, H.; Mohammad, H.; Ghaiaty, A.; Seleem, M.; Mayhoub, A. S.* Investigating the Antibacterial Activity of Biphenylthiazoles Against Methicillin- and Vancomycin-Resistant Staphylococcus aureus (MRSA and VRSA) J. Med. Chem. 2017, 60, 4074–4085.
Mohammad, H.; Younis, W.; Ezzat, H. G.; Peters, C. E.; AbdelKhalek, A.; Cooper, B.; Pogliano, K.; Pogliano, J.; Mayhoub, A. S.;* Seleem, M. Bacteriological Profiling of Diphenylureas as a Novel Class of Antibiotics. PLoS One, 2017, 12, e0182821.
Islam, E; Elsebaei, M; Mohammad, H.; Hagra, M.; Peters, E. C.; Hegazy, A. Y.; Cooper, B.; Pogliano, P., Pogliano, J.; Abulkhair, H.; Seleem, M.; Mayhoub, A. S.* Arylthiazoles Antibiotics for Targeting Intracellular Methicillin-Resistant Staphylococcus aureus (MRSA) Interfere with Bacterial Cell Wall Synthesis Eur. J. Med. Chem. 2017, 139, 665–673.
Eldesouky, H.; Mayhoub, A. S.; Hazbun, T.; Seleem, M. Reversal of azole resistance in Candida albicans by sulfa antibacterial drugs Antimicrob. Agents Chemother. 2018, 62, 701–717.
Hagras, M.; Hegazy, Y.; Elkabbany, H.; Mohammad, H.; Seleem, M.; Mayhoub, A. S.* Biphenylthiazoles Antibiotics with Oxadiazole Linker: An Approach to Improve the Physicochemical Properties Eur. J. Med. Chem. 2018, 143, 1448–1456.
Elsebaei, M; Ouf, M.; Mohammad, H.; Hegazy, Y.; Ghiaty, A.; Chen, L.; Malwal, S.; Zhang, J.; Abutaleb, N.; Oldfield, E.; Seleem, M.; and Mayhoub, A. S.* Phenylthiazols with Alkynyl Lipophilic Tail: Bacteriological Profiling and Target Identification of New Series of Anti-Methicillin-Resistant Staphylococcus aureus Eur. J. Med. Chem. 2018, 148, 195–209.
Kotb, M; Abutaleb, N.; Adel, M.; Hagras, M.; Mohammad, H.; Bayoumi, A.; Ghiaty, A.; Seleem, M.; and Mayhoub, A. S.* Phenylthiazoles with tert-Butyl Side Chain: Metabolically Stable with Anti-Biofilm Activity. Eur. J. Med. Chem. 2018, 151, 110–120.
Eslam B. Elkaeed, Jing An†, and André M. Beauchemin, Synthesis of Indazolones via Friedel–Crafts Cyclization of Blocked (Masked) N-Isocyanates, J. Org. Chem., 2017, 82 (18), pp 9890–9897.
Ngo, H.; Green, K.; Gajadeera, C.; Willby, M.; Holbrook, S.; Hou, C.; Garzan, A.; Mayhoub, A. S; Posey, J.; Tsodikov, O.; Garneau-Tsodikova, S. Potent 1,2,4-triazino[5,6b]indole-3-thioether inhibitors of the kanamycin resistance enzyme Eis from Mycobacterium tuberculosis ACS Infect Dis. 2018, 4, 1030–1040.
ElAwamy, M.; Mohammad, H.; Hussien, A.; Hagras, M.; Taha, A.; Abuzeid, K.; Seleem, M.; Mayhoub, A. S.* Alkoxyphenylthiazoles with Broad-Spectrum Activity Against Multi-Drug Resistant Gram-Positive Bacterial Pathogens Eur. J. Med. Chem. 2018, 152, 318–328.
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